Additionally,carboxylic acid derivatives containing heterocycles, N-protected amino acids,and protic functionality can be coupled in 23−96% yield with a range ofsterically hindered, electron-rich, and ...

Chemistry of Heterocycles & Natural Product Research Laboratory, Department of Chemistry, School of Advanced Sciences, Vellore Institute of Technology, Vellore 632 014, Tamil Nadu, India ...

We herein report a copper-catalyzed 1,3-aminocyclization of cyclopropanes as a direct and versatile entry into important heterocycles. This reaction was initiated by a copper-catalyzed, NFSI-promoted ...

Heterocycles found in numerous drugs could be modified more easily and directly through this method. This discovery, which allows one atom to be changed at a time without having to rebuild the whole ...

Heterocycles, like furans and pyrroles, play a vital role in drug design owing to their unique electronic properties that can enable precise interactions with biological targets. ‘[The new reaction] ...